Bifeprunox
CAS No. : 350992-10-8
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| Cat. No. : | HY-14547 |
| M.Wt: | 385.46 |
| Formula: | C24H23N3O2 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Bifeprunox is a potent dopamine D2-like and 5-HT1A receptor partial agonist with pKis of 7.19 and 8.83 for cortex 5-HT1A and striatum D2, and a pEC50 of 6.37 for hippocampus 5-HT1A, respectively. Bifeprunox is an antipsychotic for the research of schizophrenia[1][2].
IC50 & Target: pKi: 7.19 (cortex 5-HT1A) and 8.83 (striatum D2)[2]
pEC50: 6.37 (hippocampus 5-HT1A)[2]
In Vitro: Bifeprunox has a pKi of 8 at h5-HT1A receptors, with an Emax of 70%[1].
In Vivo: Bifeprunox (0.001-2.5 mg/kg) reduces marble burying in mice[2].
Bifeprunox (4-250 μg/kg) influences nicotine-seeking behaviour in response to drug-associated stimuli in rats[3].
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