Amelubant
CAS No. : 346735-24-8
(Synonyms: BIIL 284)
| Size | Price | Stock |
|---|---|---|
| 5mg | $480 | In-stock |
| 10mg | $800 | In-stock |
| 25mg | $1550 | In-stock |
| 50mg | $2400 | In-stock |
| 100mg | $3600 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-19304 |
| M.Wt: | 538.63 |
| Formula: | C33H34N2O5 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
Amelubant (BIIL 284) is a potent, oral and long acting LTB4 receptor antagonist, negligibly binds to LTB4 receptor, with Kis of 221 nM and 230 nM in vital cells and membranes. Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315. Anti-inflammatory activity[1]. IC50 & Target: Ki: 221 nM (LTB4 receptor, in vital human granulocytes), 230 nM (LTB4 receptor, in cell membranes)[1] In Vitro: Amelubant is a prodrug of active metabolites BIIL 260 and BIIL 315, which are reversible and competitive LTB4 receptor antagonists, with Kis of 1.4, 1.1 nM and 1.7, 1.9 nM in vital cells and membranes, respectively[1].
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