Bragsin2
CAS No. : 342795-08-8
| Size | Price | Stock |
|---|---|---|
| 5mg | $70 | In-stock |
| 10mg | $110 | In-stock |
| 25mg | $220 | In-stock |
| 50mg | $350 | In-stock |
| 100mg | $560 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-111550 |
| M.Wt: | 289.16 |
| Formula: | C11H6F3NO5 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
Bragsin2 is a potent, selective and noncompetitive nucleotide exchange factor BRAG2 inhibitor, with an IC50 of 3 μM. Bragsin2 binds at the interface between the PH domain of BRAG2 and the lipid bilayer, leads BRAG2 unable to activate lipidated Arf GTPase. Bragsin2 affects breast cancer stem cells[1].
IC50 & Target: IC50: 3 μM (BRAG2)[1]
In Vitro: Bragsin2 (50 μM) inhibits Arf GTPase activation in HeLa cells[1].
Bragsin2 (50 μM) inhibits the growth of SUM149 and S68, with no effect on SUM159, which lacks adhesion molecules such as integrins and cadherins[1].
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