Pirenzepine (dihydrochloride)
CAS No. : 29868-97-1
(Synonyms: LS 519; Pirenzepin (dihydrochloride); Gastrozepin (dihydrochloride))
| Size | Price | Stock |
|---|---|---|
| 100mg | $40 | In-stock |
| 500mg | $90 | In-stock |
| 1g | $162 | In-stock |
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| Cat. No. : | HY-17037 |
| M.Wt: | 424.32 |
| Formula: | C19H23Cl2N5O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 25 mg/mL (ultrasonic);H2O : 50 mg/mL (ultrasonic) |
Pirenzepine (LS 519) dihydrochloride is a selective M1 mAChR (muscarinic acetylcholine receptor) antagonist. Pirenzepine dihydrochloride reduces gastric acid secretion and reduces muscle spasm, can be used in peptic ulcers research. Pirenzepine dihydrochloride shows anti-proliferative activity to cancer cells[1][2].
In Vitro: Pirenzepine (100-140 μg/mL; 24 h) inhibits PC-3 cell proliferation activity[2].
Pirenzepine (110 μg/mL; 24 h) inhibits prostate and lung cancer cell migration[2].
Pirenzepine (100-130 μg/mL; 0-24 h) inhibits the expression of GLI1 in PC-3 cells[2].
In Vivo: Pirenzepine (intraperitoneal injection; 0.3?mg/kg; once) treatment shows beneficial effects in lipopolysaccharide-induced septic shock[3].
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