Gimatecan
CAS No. : 292618-32-7
(Synonyms: ST1481)
| Size | Price | Stock |
|---|---|---|
| 5mg | $100 | In-stock |
| 10mg | $160 | In-stock |
| 25mg | $300 | In-stock |
| 50mg | $485 | In-stock |
| 100mg | $780 | In-stock |
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| Cat. No. : | HY-B0063 |
| M.Wt: | 447.48 |
| Formula: | C25H25N3O5 |
| Purity: | >98 % |
| Solubility: | DMSO : 33.33 mg/mL (ultrasonic;warming;adjust pH to 10 with NaOH;heat to 60°C) |
Gimatecan (ST1481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity[1].
In Vitro: Gimatecan (3 to 300 ng/mL) significantly inhibits the growth of human bladder cancer models (HT1376 and MCR), thus reflecting antiproliferative potency[1].
Gimatecan causes a persistent S-phase arrest At 0.003 µg/mL and the number of S-phase cells increased after treatment with a higher concentration (0.03 µg/mL)[1].
In Vivo: Gimatecan (2 mg/kg; treatment per os, every fourth day for four times) is effective for inhibiting tumor growth[1].
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