DPC423
CAS No. : 292135-59-2
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| Cat. No. : | HY-11090A |
| M.Wt: | 568.97 |
| Formula: | C25H21ClF4N4O3S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
DPC423 is a selective and orally active factor Xa inhibitor with a Kis of 0.15 (human) and 0.3 (rabbit) nM. DPC423 exhibits Kis of 60, 61 and 6000 nM against human trypsin, plasma kallikrein and thrombin. DPC423 blocks the formation of prothrombinase complex, reduces thrombin production, inhibits fibrin formation and platelet activation. DPC423 can be used for the study of anticoagulation of arterial thrombosis[1][2].
In Vivo:DPC423 (0.08-2.5 mg/kg, i.v., for 90 min) increases blood flow in the carotid artery with an ED50 of 0.6 mg/kg[1][2].
DPC423 (1-10 mg/kg, p.o., single dose) exhibits a dose-dependent anti-thrombotic effect[1][2].
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