Iperoxo
CAS No. : 247079-84-1
| Size | Price | Stock |
|---|---|---|
| 5mg | $135 | In-stock |
| 10mg | $216 | In-stock |
| 25mg | $432 | In-stock |
| 50mg | $650 | In-stock |
| 100mg | $972 | In-stock |
| 500mg | $1944 | In-stock |
| 1 g | Get quote | |
| 5 g | Get quote | |
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| Cat. No. : | HY-122743 |
| M.Wt: | 324.16 |
| Formula: | C10H17IN2O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 62.5 mg/mL (ultrasonic;warming;heat to 60°C) |
Iperoxo is a potent superagonist of muscarinic acetylcholine receptor (mAChR) that activates M1, M2 and M3 receptors with pEC50 of 9.87, 10.1 and 9.78. Iperoxo can be used for direct probing activation-related conformational transitions of muscarinic receptors when labeled with tritium[1][2].
In Vitro:Iperoxo (0.1 nM-10 μM) activates muscarinic receptor, causes downstream signaling pathway responses, leads to phosphoinositide generation, calcium ion mobilization, and ERK1/2 phosphorylation[3].
In Vivo:Iperoxo (0.01 mg/kg, sc, single dose) exhibitis analgesic activity in rats with an ID50 of 1 μg/kg[4].
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