L-798106
CAS No. : 244101-02-8
(Synonyms: CM9; GW671021)
| Size | Price | Stock |
|---|---|---|
| 5mg | $130 | In-stock |
| 10mg | $205 | In-stock |
| 25mg | $420 | In-stock |
| 50mg | $675 | In-stock |
| 100mg | $1080 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-15274 |
| M.Wt: | 536.44 |
| Formula: | C27H22BrNO4S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
L-798106 is potent and highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM), it also has ?micromolar activities at the EP4, EP1 and EP2 receptors with Ki values of 916 nM, >5000 nM and >5000 nM, respectively[1].
IC50 & Target:Ki values: 0.3 nM (EP3 receptor); 916 nM (EP4 receptor); > 5000 nM (EP1/2 receptor)[1]
In Vitro: L-798106 (200 nM) inhibits electrical field stimulation-induced contractile responses[2].
L-798106 (10 μM) inhibits electrical field stimulation-evoked ACh release[2].
In Vivo: L-798106 (oral gavage; 50 and 100 μg/kg; once daily; 8 w) suppresses systemic insulin resistance and AT inflammation in db/db mice[3].
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