U-101958 (maleate)
CAS No. : 224170-09-6
(Synonyms: PNU-101958 (maleate))
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| Cat. No. : | HY-123663 |
| M.Wt: | 455.55 |
| Formula: | C25H33N3O5 |
| Purity: | >98 % |
| Solubility: |
U-101958 (PNU-101958) maleate is a highly selective ligand and antagonist for dopamine D4 receptor, with an IC50 of 2.7 nM. U-101958 maleate behaves as an agonist in HEK-293 cells expressing the human recombinant D4.4 receptor. U-101958 maleate is an antipsychotic[1][2].
In Vitro:U-101958 inhibits Forskolin (HY-15371)-stimulated cyclic AMP accumulation in HEK293/D4 cells in a concentration-dependent way[1].
[3H]PNU-101958 is a D4 receptor probe. [3H]PNU-101958 binding sites in non-human primate brain appear to reflect D4 dopamine receptor distribution[2].
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