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|---|---|---|
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| 500 mg | Get quote | |
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| Cat. No. : | HY-119938 |
| M.Wt: | 563.69 |
| Formula: | C34H37N5O3 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Tuberculosis inhibitor 1 is a potent and non-cytotoxic trypanosoma brucei growth inhibitor with an EC50 of 5 nM[1]. IC50 & Target: EC50: 5 nM (Trypanosoma brucei)[1] In Vitro: Tuberculosis inhibitor 1 is selective over other parasites, such as Trypanosoma cruzi and Plasmodium falciparum (T. cruzi EC50 8120 nM, P. falciparum EC50 3624 nM)[1].
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