Crobenetine
CAS No. : 221019-25-6
(Synonyms: BIII-890; BIII-890 CL (free acid))
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| Cat. No. : | HY-16923 |
| M.Wt: | 379.54 |
| Formula: | C25H33NO2 |
| Purity: | >98 % |
| Solubility: |
Crobenetine (BIII-890), a benzomorphan derivative, is a potent, selective, and highly use-dependent Na+ channel blocker. Crobenetine displaces [3H]BTX from site 2 of the Na+ channel (IC50=49 nM) in rat brain synaptosomes, yet exhibits only low binding affinity for other receptors and ion channels. Crobenetine protects brain tissue from the deleterious effects of focal cerebral ischemia in rodents[1]. In Vivo:Crobenetine (BIII-890; BIII 890 CL; 3-30 mg/kg; s.c.) reduces lesion size in mice and rats when administered 5 min after permanent focal cerebral ischemia at doses that does not impair motor coordination[1].
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