GYKI-47261
CAS No. : 220445-20-5
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| Cat. No. : | HY-19435 |
| M.Wt: | 322.79 |
| Formula: | C18H15ClN4 |
| Purity: | >98 % |
| Solubility: |
GYKI-47261 is a competitive, orally active, and selective AMPA receptor antagonist with an IC50 of 2.5 μM. GYKI-47261 has broad spectrum anticonvulsive activity and neuroprotective effects. GYKI-47261 is also a potent inducer of CYP2E1[1][2].
In Vivo:GYKI-47261 (6 mg/kg; i.v.) shows antiischemice effect in a transient focal ischemia model, in rats. GYKI-47261 (p.o.) potently mitigated the tremor induced by oxotremorine with ED50 of 16.8 mg/kg in male CD1 mice[1].
GYKI-47261(20 mg/kg; i.p.) reverses the dopamine depleting effect of MPTP[1].
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