N-Pentanoyl 2-benzyltryptamine
CAS No. : 220339-00-4
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| Cat. No. : | HY-107628 |
| M.Wt: | 334.45 |
| Formula: | C22H26N2O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
N-Pentanoyl 2-benzyltryptamine is a potent and selective antagonist of MT2 melatonin receptor, with a pKi of 8.03 for human MT2. N-Pentanoyl 2-benzyltryptamine shows 89- and 229-fold selectivity for human MT2 over human mt1 and Xenopus mel1c receptor subtypes. N-Pentanoyl 2-benzyltryptamine can inhibit melatonin-induced enhancement of electrically-evoked responses[1][2].
In Vitro: N-Pentanoyl 2-benzyltryptamine (compound 9) (0.1-100 μM; 2 h) antagonizes pigment aggregation induced by melatonin (10 nM) in Xenopus laevis melanophores[1].
N-Pentanoyl 2-benzyltryptamine has no agonist activity at concentrations up to 100 μM[1].
N-Pentanoyl 2-benzyltryptamine (60 nM) significantly alteres the potency of melatonin in the rat tail artery at low concentrations of the MT2 selective ligands, with a pEC50 of 8.83[2].
N-Pentanoyl 2-benzyltryptamine (5 μM) causes a significant rightward displacement of the vasoconstrictor effect of melatonin at concentrations non-selective for mt1 and MT2 receptors[2].
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