BI-2545
CAS No. : 2162961-71-7
| Size | Price | Stock |
|---|---|---|
| 5mg | $95 | In-stock |
| 10mg | $140 | In-stock |
| 25mg | $250 | In-stock |
| 50mg | $375 | In-stock |
| 100mg | $560 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-124772 |
| M.Wt: | 527.42 |
| Formula: | C23H19F6N5O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
BI-2545 is a potent autotaxin (ATX) inhibitor that significantly reduces LPA, with IC50s of 2.2 nM and 3.4 nM for human ATX and rat ATX, respectively[1].
IC50 & Target: C50: 2.2 nM (human ATX), 3.4 nM (rat ATX)[1]
In Vitro: BI-2545 displays good potency in the LPA and rat whole blood assay with IC50s of 29 nM and 96 nM, respectively[1].
In Vivo: BI-2545 (10 mg/kg; p.o.) has high and sustained in vivo efficacy in reducing LPAs[1].
BI-2545 (10 mg/kg; p.o.) has a half-life of t1/2=3.4 hours[1].
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- Cat. No.:
- HY-124772
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