CLK-IN-T3
CAS No. : 2109805-56-1
| Size | Price | Stock |
|---|---|---|
| 5mg | $120 | In-stock |
| 10mg | $210 | In-stock |
| 25mg | $390 | In-stock |
| 50mg | $680 | In-stock |
| 100mg | $1150 | In-stock |
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| Cat. No. : | HY-115470 |
| M.Wt: | 482.58 |
| Formula: | C28H30N6O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 4.83 mg/mL (ultrasonic;warming) |
CLK-IN-T3 is a high potent, selective, and stable CDC-like kinase (CLK) inhibitor with IC50s of 0.67 nM, 15 nM, and 110 nM for CLK1, CLK2, and CLK3 protein kinases, respectively. CLK-IN-T3 has anti-cancer activity[1].
In Vitro: CLK-IN-T3 inhibits DYRK1A (IC50=260 nM) and DYRK1B (IC50=230 nM)[1].
CLK-IN-T3 (0.1-10.0 µM; 24 hours) results in mild cell cycle arrest at the G2/M boundary with long-duration (24 h)[1].
CLK-IN-T3 (0.5-1.0 µM; 6 hours) decreases phosphorylation of CLK-targeted SR proteins and CLK proteins increase slightly[1].
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