PD 168568
CAS No. : 210688-56-5
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| Cat. No. : | HY-103407 |
| M.Wt: | 349.47 |
| Formula: | C22H27N3O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
PD 168568 is a orally active and potent dopamine receptor D4 (DRD4) antagonist. PD 168568 contains an isoindolinone and is selective for the D4 receptor versus D2 and D3, with Ki values of 8.8, 1842, and 2682 nM, respectively. PD 168568 can be used for glioblastoma (GBM) research[1][2]. In Vitro:PD 168568 shows selectivity inhibition toward glioblastoma neural stem cells (GNS), with IC50 of 25-50 µM[1]. In Vivo:PD 168568 (3 mg/kg, Oral) has ability to inhibit amphetamine-stimulated locomotor activity in the rat[3].
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