GSK-LSD1 (dihydrochloride)
CAS No. : 2102933-95-7
| Size | Price | Stock |
|---|---|---|
| 1mg | $45 | In-stock |
| 5mg | $96 | In-stock |
| 10mg | $144 | In-stock |
| 25mg | $288 | In-stock |
| 50mg | $450 | In-stock |
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| Cat. No. : | HY-100546A |
| M.Wt: | 289.24 |
| Formula: | C14H22Cl2N2 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 62.5 mg/mL |
GSK-LSD1 dihydrochloride is a potent, selective and irreversible lysine specific demethylase 1 (LSD1) inhibitor with an IC50 of 16 nM. IC50 & Target: IC50: 16 nM (LSD1)[1] In Vitro: GSK-LSD1 shows more than 1000 fold selectivity over other closely related FAD utilizing enzymes including LSD2, and monoamine oxidases MAO-A, MAO-B[1]. GSK-LSD1 can inhibit KDM1A/LSD1 enzyme activity. GSK-LSD1 induces the formation of LC3-II in U2OS cells. The electronic microscopy shows the formation of autophagosome with GSK-LSD1 treatment. GSK-LSD1 potently inhibits proliferation of varies cancer cell lines by changing gene expression patterns[2].
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