PI3Kα-IN-1
CAS No. : 2100855-80-7
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| Cat. No. : | HY-124647 |
| M.Wt: | 483.52 |
| Formula: | C26H25N7O3 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
PI3Kα-IN-1 is a PI3Kα inhibitor (IC50 < 0.5 nM), and also inhibits mTOR (IC50: 104 nM)[1].
In Vitro:PI3Kα-IN-1 shows good stability in the mouse liver microsome assay (t1/2 values > 60 minutes)[1].
PI3Kα-IN-1 (48 h) induces cytotoxicity in MDC7 cells with an IC50 value of around 170 nM[1].
PI3Kα-IN-1 (15-250 nM) inhibits phospho4EBP, phosphor-P70SK6 and phospho-473AKT in MCF7 cells[1].
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