AZ3451
CAS No. : 2100284-59-9
| Size | Price | Stock |
|---|---|---|
| 5mg | $77 | In-stock |
| 10mg | $132 | In-stock |
| 25mg | $297 | In-stock |
| 50mg | $517 | In-stock |
| 100mg | $902 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-112558 |
| M.Wt: | 571.46 |
| Formula: | C30H27BrN4O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
AZ3451 is a potent protease-activated receptor-2 (PAR2) antagonist with IC50 of 23 nM. IC50 & Target: Protease-activated receptor-2 (IC50= 23 nM)[1] In Vitro: Antagonist AZ3451 binds to a remote allosteric site outside the helical bundle of the protease-activated receptor 2. AZ3451 is highly lipophilic, which coincides with the hydrophobic nature of the binding pocket within the membrane. Antagonist binding prevents structural rearrangements required for receptor activation and signalling[1].
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