| Size | Price | Stock |
|---|---|---|
| 5mg | $550 | In-stock |
| 10mg | $850 | In-stock |
| 25mg | $1850 | In-stock |
| 50mg | $2775 | In-stock |
| 100mg | $4000 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-103633 |
| M.Wt: | 871.90 |
| Formula: | C44H45N11O9 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 50 mg/mL |
PROTAC BET Degrader-1 is a PROTAC connected by ligands for Cereblon and BET, decreasing BRD2, BRD3, and BRD4 protein levels at low concentration. IC50 & Target:BET[1] In Vitro: PROTAC BET Degrader-1 (Compound 9) is a potent BET degrader based on PROTAC, decreases the level of BRD2, BRD3, and BRD4 proteins in RS4;11 cells at 3-10 nM, and inhibits the growth of this cell line with an IC50 of 4.3 nM, and 45.5 nM for MOLM-13 cells[1].
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