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|---|---|---|
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| Cat. No. : | HY-120924 |
| M.Wt: | 485.42 |
| Formula: | C23H21F6N3O2 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
BRD9185 is a Dihydroorotate dehydrogenase (DHODH) inhibitor, with an EC50 of 16 nM against multidrug-resistant blood-stage parasites in vitro and is curative after just three doses in a P. berghei mouse model[1]. IC50 & Target: EC50: 16 nM (DHODH in vitro)[1].
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