CCG 224061
CAS No. : 2055990-82-2
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| Cat. No. : | HY-120718 |
| M.Wt: | 325.39 |
| Formula: | C19H20FN3O |
| Purity: | >98 % |
| Solubility: |
CCG 224061 is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with a IC50 of 0.066 μM. CCG 224061 inhibits GRK activity in cardiomyocytes[1]. CCG 224061 is applicable to research related to heart disease, heart failure, myocardial hypertrophy and hypertension[1][2].
In Vitro:CCG 224061 (E18) potently and selectively inhibits GRK2 with an IC50 of 0.07 μM, while it shows weak inhibitory effects on GRK5 (IC50 12.8 μM) and GRK1 (IC50 65.7 μM)[1].
CCG 224061 (5 min) potently inhibits GRK2 (IC50 = 0.066 μM) and exhibits activity against GRK1 (IC50 = 6.4 μM), GRK5 (IC50 = 1.3 μM), PKA (IC50 = 3.1 μM) and ROCK1 (100% inhibition at 10 μM) in in vitro purified kinase assays[2].
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