MZP-54
CAS No. : 2010159-47-2
| Size | Price | Stock |
|---|---|---|
| 1mg | $220 | In-stock |
| 5mg | $496 | In-stock |
| 10mg | $744 | In-stock |
| 25mg | $1400 | In-stock |
| 50 mg | Get quote | |
| 100 mg | Get quote | |
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| Cat. No. : | HY-112376 |
| M.Wt: | 1036.67 |
| Formula: | C55H66ClN7O9S |
| Purity: | >98 % |
| Solubility: | Ethanol : 50 mg/mL (ultrasonic) |
MZP-54 is a PROTAC connected by ligands for von Hippel-Lindau and BRD3/4, with a Kd of 4 nM for Brd4BD2. IC50 & Target:Kd: 4 nM (Brd4BD2)[1] In Vitro: MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology, with a Kd of 4 nM for Brd4BD2. MZP-54 binds to VHL-EloC-EloB protein (VCB) with a Kd of 105 ± 24 nM. MZP-54 shows an inhibitory activity against MV4;11 and HL60 cells, with pEC50s of 7.08 ± 0.05 and 6.37 ± 0.03, respectively. MZP-54 also exhibits high depletion of cMyc levels[1].
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