Thermopsoside
CAS No. : 19993-32-9
| Size | Price | Stock |
|---|---|---|
| 1mg | $112 | In-stock |
| 5mg | $280 | In-stock |
| 10mg | $420 | In-stock |
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| 100 mg | Get quote | |
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| Cat. No. : | HY-N6023 |
| M.Wt: | 462.40 |
| Formula: | C22H22O11 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Thermopsoside is a CYP450 isoenzyme inhibitor and PXR activator. Thermopsoside inhibits CYP3A4, CYP2C19, CYP2D6 and CYP2C9 with IC50 values of 6.0 μM, 9.5 μM, 12.0 μM and 32.0 μM, respectively[1].
In Vitro:Thermopsoside (0.3-30 μM; 48 h) activates PXR but exerts only marginal effects on the mRNA expression of CYP3A4, CYP1A2, CYP2C9, and P-gp in transiently transfected HepG2 cells[1].
Thermopsoside (100 μM; 10 min pre-incubation, 1 h with calcein-AM) does not inhibit P-glycoprotein activity in hMDR1-MDCK-II cells at 100 μM[1].
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