CGP71683 hydrochloride
CAS No. : 192322-50-2
(Synonyms: CGP71683A)
| Size | Price | Stock |
|---|---|---|
| 5mg | $133 | In-stock |
| 10mg | $200 | In-stock |
| 25mg | $337 | In-stock |
| 50mg | $470 | In-stock |
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| 200 mg | Get quote | |
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| Cat. No. : | HY-107723 |
| M.Wt: | 512.07 |
| Formula: | C26H30ClN5O2S |
| Purity: | >98 % |
| Solubility: | DMSO : 160 mg/mL (ultrasonic) |
CGP71683 hydrochloride is a competitive neuropeptide Y5 receptor antagonist with a Ki of 1.3 nM, and shows no obvious activity at Y1 receptor (Ki, >4000 nM) and Y2 receptor (Ki, 200 nM) in cell membranes. IC50 & Target: Ki: 1.3 nM (Y5 receptor), 200 nM (Y2 receptor), >4000 nM (Y1 receptor)[1] In Vitro: CGP71683 hydrochloride is a competitive neuropeptide Y5 receptor antagonist with a Ki of 1.3 nM, and shows no obvious activity at Y1 receptor (Ki, >4000 nM) and Y2 receptor (Ki, 200 nM) in cell membranes[1]. In Vivo: CGP71683 (15 nmol/rat, icv, twice daily) shows anorexigenic effect, reducing food intake and bady weight of fed rats. CGP71683 causes 3-times higher serum total T4 and 37% increase in free T4 in the fasted rats than in the fasted controls rats[2].
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