GGTI-2133
CAS No. : 191102-79-1
| Size | Price | Stock |
|---|---|---|
| 1mg | $300 | In-stock |
| 5mg | $750 | In-stock |
| 10mg | $1150 | In-stock |
| 25mg | $1900 | In-stock |
| 50mg | $2750 | In-stock |
| 100mg | $3850 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-12369 |
| M.Wt: | 456.54 |
| Formula: | C27H28N4O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
GGTI-2133, a peptidomimetic, is a selective geranylgeranyltransferase I (GGTase-I) inhibitor with an IC50 of 38 nM. GGTI-2133 shows 140-fold selectivity over farnesyltransferase (FTase) (IC50 of 5.4 μM). GGTI-2133 inhibits the geranylation of Rap-1A with an IC50 of 10 μM. GGTI-2133 can be used for the study of eosinophilic airway inflammation such as asthma[1][2]. IC50 & Target:Geran ylgeranyltransferase (GGTase) In Vivo:GGTI-2133 (5 mg/kg; intraperitoneal injection; once a day; for 10 days) inhibits infiltration of inflammatory cells into airways in mouse experimental asthma[2].
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