Bremelanotide
CAS No. : 189691-06-3
(Synonyms: PT-141)
| Size | Price | Stock |
|---|---|---|
| 5mg | $42 | In-stock |
| 10mg | $66 | In-stock |
| 25mg | $132 | In-stock |
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| Cat. No. : | HY-18678 |
| M.Wt: | 1025.16 |
| Formula: | C50H68N14O10 |
| Purity: | >98 % |
| Solubility: | H2O : 100 mg/mL (ultrasonic) |
Bremelanotide (PT-141) is a melanocortin receptor agonist. Bremelanotide can activate MC4R and increases dopamine release. Bremelanotide induces appetitive sexual behaviors, female mounting behavior, and repetitive self-grooming. Bremelanotide can be used for the research of hypoactive sexual desire disorders[1][2][3].
In Vitro:Bremelanotide (10−3-105 nM) binds to MC3R and MC4R in a concentration-dependent manner[3].
Bremelanotide induces cAMP accumulation in cell-free assays with EC50 values of 0.4 nM for MC3R and 0.2 nM for MC4R[3].
In Vivo:Bremelanotide (50-200 μg/kg; s.c.) selectively increases appetitive sexual behaviors (solicitations, hops and darts) in hormone-primed ovariectomized female rats via activation of MC4R and dopamine release in the medial preoptic area[1].
Bremelanotide (0.01-10 mg/kg; i.p.; single dose) induces dose-dependent repetitive grooming behavior in male and female mice, with 1 mg/kg being the lowest effective grooming dose that does not cause anxiety-like behavior[2].
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