CL 316243 (free acid)
CAS No. : 183720-02-7
| Size | Price | Stock |
|---|---|---|
| 5mg | $170 | In-stock |
| 10mg | $252 | In-stock |
| 25mg | $420 | In-stock |
| 50mg | $670 | In-stock |
| 100mg | $1070 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-116771 |
| M.Wt: | 421.83 |
| Formula: | C20H20ClNO7 |
| Purity: | >98 % |
| Solubility: |
CL316243 free acid is a highly potent selective β3-adrenoceptor agonist with a EC50 of 3 nM, but is an extremely poor to β1/2- receptors. CL316243 free acid is a effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate. CL316243 free acid has the potential for the treatment obesity, diabetes and urge urinary incontinence[1][2][3]. In Vitro:CL 316243 free acid displays binding affinities with IC50 values of 0.6 μM and 1 μM for rat heart and rat soleus muscle respectively[1]. CL 316243 free acid inhibits spontaneously contracting, isolated rat detrusor strips in a concentration dependent manner with a mean concentration inhibiting 50% of maximal response of 2.65 nM[3]. In Vivo:CL316243 free acid (subcutaneously injection; 0.1 mg/kg/day; once a day; 1 weeks) elevates the mRNA and protein expression levels of UCP1 in BAT, irrespective of diet[2].
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