Valemetostat
CAS No. : 1809336-39-7
(Synonyms: DS-3201)
| Size | Price | Stock |
|---|---|---|
| 1mg | $119 | In-stock |
| 5mg | $250 | In-stock |
| 10mg | $420 | In-stock |
| 25mg | $695 | In-stock |
| 50mg | $990 | In-stock |
| 100mg | $1310 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-109108 |
| M.Wt: | 488.02 |
| Formula: | C26H34ClN3O4 |
| Purity: | >98 % |
| Solubility: | DMSO : 70 mg/mL (ultrasonic) |
Valemetostat (DS-3201), a first-in-class EZH1/2 dual inhibitor with IC50 values ＜10 nM. Valemetostat can be used for the research of relapsed/refractory peripheral T-cell lymphoma[1][2][3]. IC50 & Target:IC50: ＜10 nM (EZH1/2)[3] In Vitro:Valemetostat (1-1000 nM) strongly and specifically inhibits EZH1 and EZH2 with IC50 values ＜10 nM[3]. Valemetostat (100 nM; 7 d) effectively removes H3K27me3 and also prevents unexpected gain of H3K27me3[3]. Valemetostat (0.1-100 nM; 7 d) potently inhibits H3K27me3 by low-dose treatment in the sensitive lymphoma types[3]. In Vivo:Valemetostat (0.01 mg/g; i.p.; once) prevents the changes of H3K27me3 after exercise training[2].
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