PSB-12379
CAS No. : 1802226-78-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $204 | In-stock |
| 10mg | $312 | In-stock |
| 25mg | $672 | In-stock |
| 50 mg | Get quote | |
| 100 mg | Get quote | |
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| Cat. No. : | HY-100747 |
| M.Wt: | 515.35 |
| Formula: | C18H23N5O9P2 |
| Purity: | >98 % |
| Solubility: | H2O : 125 mg/mL (ultrasonic) |
PSB-12379, a nucleotide analogue, is a potent Ecto-5'-Nucleotidase (CD73) inhibitor with Kis of 9.03 nM (rat) and 2.21 nM (human)[1][2]. IC50 & Target:Ki: 9.03 nM (rat), 2.21 nM (human) (Ecto-5’-Nucleotidase)[1] In Vitro: Metabolism: Only a small percentage (<23%) of PSB-12379 (10g) is metabolized under the applied conditions, while >77% of the compounds are recovered unchanged after a long incubation for 8 h. PSB-12379 (10g) is somewhat less stable, and 56% are metabolized within 8 h. Hydrolytic cleavage of the glycosidic bond, which is a typical phase I reaction of nucleosides and nucleotides, was observed as the main reaction[1].
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