Eptapirone
CAS No. : 179756-58-2
(Synonyms: F 11440)
| Size | Price | Stock |
|---|---|---|
| 5mg | $56 | In-stock |
| 10mg | $93 | In-stock |
| 25mg | $187 | In-stock |
| 50mg | $300 | In-stock |
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| Cat. No. : | HY-19946 |
| M.Wt: | 345.40 |
| Formula: | C16H23N7O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
Eptapirone (F11440) is a potent, selective and orally active 5-HT1A receptor agonist (pKi = 8.33). Eptapirone can inhibit cAMP production. Eptapirone can reduce 5-HT levels and increase corticosterone levels. Eptapirone shows potent anxiolytic and antidepressant potential. Eptapirone can be used for the research of neurological disease, such as anxiety and depression[1].
In Vitro:Eptapirone decreases the Forskolin (HY-15371)-induced stimulation of cAMP with an pEC50 value of 6.8 in HeLa cells[1].
In Vivo:Eptapirone (0.16-640 mg/kg, p.o., a single dose) produces anxiolytic- and antidepressant-like effects in anxiety and depression rats models[1].
Eptapirone (0.01-0.63 mg/kg, i.p.) reduces 5-HT levels in microdialysates from the ventral hippocampus of rats[1].
Eptapirone (0.0063-160 mg/kg, p.o.) increases plasma corticosterone levels in rats[1].
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