Src Inhibitor 1
CAS No. : 179248-59-0
(Synonyms: Src Kinase Inhibitor 1; Src-l1)
| Size | Price | Stock |
|---|---|---|
| 5mg | $67 | In-stock |
| 10mg | $112 | In-stock |
| 25mg | $225 | In-stock |
| 50mg | $360 | In-stock |
| 100mg | $577 | In-stock |
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| Cat. No. : | HY-101053 |
| M.Wt: | 373.40 |
| Formula: | C22H19N3O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 9.09 mg/mL (ultrasonic) |
Src Inhibitor 1 is a potent, ATP-competitive and selective dual site Src tyrosine kinase inhibitor with IC50 values of 44 nM for Src and 88nM for Lck. IC50 & Target: IC50: 44 nM (Src), 88 nM (Lck)[1] In Vitro: Src-I1 is competitive with both ATP and peptide binding sites of the kinase. The IC50 values are 44 and 88 nM for Src and Lck, respectively[1]. Src-I1, is found to be a potent inhibitor of Src (IC50=0.18 μM), but also inhibited other Src family members, such as Lck, Csk and Yes with similar potency to Src, and RIP2 (IC50=0.026 μM) with even greater potency. In addition, it inhibited CHK2 with similar potency to Src, and Aurora B with slightly lower potency[2].
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