Eletriptan (hydrobromide)
CAS No. : 177834-92-3
(Synonyms: Eletriptan HBr; UK-116044 (hydrobromide))
| Size | Price | Stock |
|---|---|---|
| 5mg | $66 | In-stock |
| 10mg | $83 | In-stock |
| 25mg | $170 | In-stock |
| 50mg | $280 | In-stock |
| 100mg | $462 | In-stock |
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| Cat. No. : | HY-A0010 |
| M.Wt: | 463.43 |
| Formula: | C22H27BrN2O2S |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
Eletriptan hydrobromide (Eletriptan HBr) is a 5-HT1B and 5-HT1D receptor agonist with antimigraine activity, with Ki of 0.92 nM and 3.14 nM, respectively[1][2][3][4][5][6]. In Vivo:Eletriptan (1-1000 μg/kg; i.v.; after a 60-minute stabilization period, dosed at 5-minute intervals with readings taken every 30 seconds) hydrobromide dose-dependently reduces carotid blood flow in anesthetized dogs[1]. Eletriptan (30-300 μg/kg; i.v.) hydrobromide dose-dependently inhibits dural plasma protein extravasation in anesthetized rats and rapidly and completely inhibits plasma protein extravasation from the dura mater at a dose of 100 μg/kg[1].
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