Estradiol 3-sulfamate
CAS No. : 172377-52-5
(Synonyms: BLE 00084; E2MATE; ES-J 995)
| Size | Price | Stock |
|---|---|---|
| 5mg | $360 | In-stock |
| 10mg | $576 | In-stock |
| 25mg | $1152 | In-stock |
| 50mg | $1840 | In-stock |
| 100mg | $2940 | In-stock |
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| Cat. No. : | HY-U00112 |
| M.Wt: | 351.46 |
| Formula: | C18H25NO4S |
| Purity: | >98 % |
| Solubility: | DMSO : 62.5 mg/mL (ultrasonic) |
Estradiol 3-sulfamate (BLE 00084; E2MATE; ES-J 995) is a potent, long-acting, and orally active steroid sulfatase inhibitor; inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. IC50 & Target: IC50: 251 nM (estrone sulfatase)[1]
Ki: 133 nM (estrone sulfatase)[1]
In Vitro: Introduction of a fluoro, chloro, or bromo moiety at the C-2 position of EMATE and Estradiol 3-sulfamate and that of a fluoro moiety at the C-4 position of the parent sulfamates markedly increase the estrone sulfatase inhibitory activity[1]. In Vivo: Estradiol 3-sulfamate is readily transformed and absorbed in the gut into its oxidative metabolite, EMATE, and both compounds have already been shown to be potent, long-acting, and orally active STS inhibitors[2].Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
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