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|---|---|---|
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| Cat. No. : | HY-123056 |
| M.Wt: | 484.42 |
| Formula: | C24H27Cl2N7 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
EAD1 is a potent autophagy inhibitor with antiproliferative activity in lung and pancreatic cancer cells. EAD1 also induces apoptosis[1].
In Vitro: EAD1 (0-200 μM; 72 hours) has antiproliferative activity against human cancer cell lines[1].
EAD1 (5-75 μM; 24 hours) induces apoptosis in the H460 cells in a concentration-dependent manner[1].
EAD1 (1-25 μM; 24 hour) increases the punctate LC3 signal in H460 cells[1].
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