LJH685
CAS No. : 1627710-50-2
| Size | Price | Stock |
|---|---|---|
| 5mg | $100 | In-stock |
| 10mg | $160 | In-stock |
| 25mg | $320 | In-stock |
| 50mg | $512 | In-stock |
| 100mg | $768 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-19712 |
| M.Wt: | 381.42 |
| Formula: | C22H21F2N3O |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 31 mg/mL |
LJH685 is a potent, ATP-competitive and selective RSK inhibitor, inhibits RSK1, 2, and 3 biochemical activities with IC50s of 6, 5, 4 nM, respectively[1]. IC50 & Target: IC50: 6 nM (RSK1), 5 nM (RSK1), 4 nM (RSK1)[1] In Vitro: LJH685 (0.01-100 μM; 72 hours) efficiently inhibits the growth of MDA-MB-231 and H358 cells in soft agar with EC50s of 0.73 and 0.79 μM, respectively[1]. LJH685 (0.1-10 μM; 4 hours) efficiently reduces phosphorylation of YB1 at submicromolar concentrations and causes nearly complete inhibition at higher concentrations[1].
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