NTRC-824
CAS No. : 1623002-61-8
| Size | Price | Stock |
|---|---|---|
| 1mg | $200 | In-stock |
| 5 mg | Get quote | |
| 10 mg | Get quote | |
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| Cat. No. : | HY-12436 |
| M.Wt: | 553.55 |
| Formula: | C25H26F3N3O6S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
NTRC-824 (Compound 5) is a potent, selective and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist with an IC50 of 38 nM and a Ki of 202 nM. NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM)[1].
IC50 & Target: IC50: 38 nM (Nurotensin receptor type 2)[1]
Ki: 202 nM (Nurotensin receptor type 2)[1]
In Vitro: Testing of NTRC-824 (Compound 5) at the NTS1 receptor shows no binding activity in the NTS1 assay up to 30 μM, making NTRC-824 (Compound 5) selective for NTS2 in both the binding and functional assays. NTRC-824 (Compound 5) is the first nonpeptide compound that behaves like, and is more active than, the endogenous ligand[1].
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Inquiry Information- Product Name:
- NTRC-824
- Cat. No.:
- HY-12436
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