Enitociclib
CAS No. : 1610408-97-3
(Synonyms: (+)-BAY-1251152; (+)-VIP152; (S)-Enitociclib)
| Size | Price | Stock |
|---|---|---|
| 2mg | $132 | In-stock |
| 5mg | $228 | In-stock |
| 10mg | $348 | In-stock |
| 25mg | $665 | In-stock |
| 50mg | $1068 | In-stock |
| 100mg | $1700 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-103019 |
| M.Wt: | 404.43 |
| Formula: | C19H18F2N4O2S |
| Purity: | >98 % |
| Solubility: | DMSO : 113.3 mg/mL (ultrasonic;warming) |
(+)-Enitociclib ((+)-BAY-1251152) is the enantiomer of Enitociclib (HY-103019E) with (+) optical rotation. Enitociclib is a selective CDK9 inhibitor and apoptosis inducer. Enitociclib inhibits CDK9 activity and reduces the phosphorylation of Ser2 in the carboxyl-terminal domain (CTD) of RNA polymerase Pol II, thereby downregulating the transcription of key oncogenes such as MYC and MCL1. Enitociclib has anti-proliferative activity targeting MYC+ lymphoma and multiple myeloma (MM) cells, and has synergistic effects with Bortezomib (HY-10227) and Lenalidomide (HY-A0003), and can be used in the research of hematological malignancies[1][2].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Enitociclib
- Cat. No.:
- HY-103019
- Quantity:
Your information is safe with us.