Bremelanotide (Acetate)
CAS No. : 1607799-13-2
(Synonyms: PT-141 Acetate)
| Size | Price | Stock |
|---|---|---|
| 5mg | $42 | In-stock |
| 10mg | $66 | In-stock |
| 25mg | $132 | In-stock |
| 50mg | $198 | In-stock |
| 100mg | $250 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-18678A |
| M.Wt: | 1085.22 |
| Formula: | C52H72N14O12 |
| Purity: | >98 % |
| Solubility: | DMSO : 125 mg/mL (ultrasonic);H2O : ≥ 50 mg/mL |
Bremelanotide (PT-141) Acetate is a melanocortin receptor agonist. Bremelanotide Acetate can activate MC4R and increases dopamine release. Bremelanotide Acetate induces appetitive sexual behaviors, female mounting behavior, and repetitive self-grooming. Bremelanotide Acetate can be used for the research of hypoactive sexual desire disorders[1][2][3].
In Vitro:Bremelanotide (10−3-105 nM) Acetate binds to MC3R and MC4R in a concentration-dependent manner[3].
Bremelanotide Acetate induces cAMP accumulation in cell-free assays with EC50 values of 0.4 nM for MC3R and 0.2 nM for MC4R[3].
In Vivo:Bremelanotide (50-200 μg/kg; s.c.) Acetate selectively increases appetitive sexual behaviors (solicitations, hops and darts) in hormone-primed ovariectomized female rats via activation of MC4R and dopamine release in the medial preoptic area[1].
Bremelanotide (0.01-10 mg/kg; i.p.; single dose) Acetate induces dose-dependent repetitive grooming behavior in male and female mice, with 1 mg/kg being the lowest effective grooming dose that does not cause anxiety-like behavior[2].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Bremelanotide (Acetate)
- Cat. No.:
- HY-18678A
- Quantity:
Your information is safe with us.