Lobradimil
CAS No. : 159768-75-9
(Synonyms: RMP 7)
| Size | Price | Stock |
|---|---|---|
| 1mg | $450 | In-stock |
| 5mg | $1100 | In-stock |
| 10mg | $1888 | In-stock |
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| 100 mg | Get quote | |
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| Cat. No. : | HY-105155 |
| M.Wt: | 1098.28 |
| Formula: | C49H75N15O12S |
| Purity: | >98 % |
| Solubility: | H2O : ≥ 50 mg/mL |
Lobradimil (RMP 7), a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). Lobradimil increases the permeability of the BBB. Lobradimil can be used in the research of brain tumors[1].
In Vitro:Lobradimil induces an increase in intracellular free calcium levels in RBME cells[3].
Lobradimil (0.01-0.5 nM, 15 min) increases the permeability of human brain microvascular endothelial cell (HMBEC) monolayers1[4].
In Vivo:Lobradimil (2.5-mg/kg bolus plus 10 mg/kg/h for 90 minutes) increases brain tumor permeability and shows hypotensive effects in RG2 glioma cells-implanted rats[2].
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