FSCPX
CAS No. : 156547-56-7
| Size | Price | Stock |
|---|---|---|
| 1mg | $230 | In-stock |
| 5mg | $580 | In-stock |
| 10mg | $870 | In-stock |
| 25mg | $1480 | In-stock |
| 50mg | $1980 | In-stock |
| 100mg | $2650 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-116042 |
| M.Wt: | 506.55 |
| Formula: | C23H27FN4O6S |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (ultrasonic;warming;heat to 60°C) |
FSCPX is a potent and selective irreversible antagonist of A1 adenosine receptor (A1AR), with low nanomolar potency for binding to the A1AR. FSCPX could modify the effect of NBTI, a nucleoside transport inhibitor, by reducing the interstitial adenosine level in the guinea pig atrium[1][2].
IC50 & Target: A1AR[1]
In Vitro: FSCPX irreversibly blocks the binding of [3H]-8-cyclopentyl-1,3dipropylxanthine ([3H]DPCPX), with an IC50 of 11.8±3.2 nM in DDT1 MF2 cells[1].
FSCPX (20 μM; 48 h) attenuates protection from necrosis and apoptosis in A1AR-overexpressing LLC-PK1 cells[3].
FSCPX (2-20 μM; 48 h) reverses the upregulation of HSP27 mRNA and protein in A1AR-overexpressing LLC-PK1 cells without an effect on the mRNA or protein for HSP70[3].
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