Dexmedetomidine (hydrochloride)
CAS No. : 145108-58-3
(Synonyms: (+)-Medetomidine (hydrochloride); (S)-Medetomidine (hydrochloride))
| Size | Price | Stock |
|---|---|---|
| 5mg | $55 | In-stock |
| 10mg | $66 | In-stock |
| 25mg | $130 | In-stock |
| 50mg | $198 | In-stock |
| 100mg | $285 | In-stock |
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| Cat. No. : | HY-17034A |
| M.Wt: | 236.74 |
| Formula: | C13H17ClN2 |
| Purity: | >98 % |
| Solubility: | H2O : ≥ 50 mg/mL;DMSO : 250 mg/mL (ultrasonic) |
Dexmedetomidine hydrochloride ((+)-Medetomidine hydrochloride) is a potent, selective and orally active agonist of α2-adrenoceptor, with a Ki of 1.08 nM. Dexmedetomidine hydrochloride shows 1620-fold selectivity against α1-adrenoceptor. Dexmedetomidine hydrochloride exhibits anxiolysis, sedation, and modest analgesia effects[1][2][3].
In Vitro:Medetomidine has high selectivity for α2-adrenoceptor, (Ki=1.08 nM) over α1 adrenoceptors (Ki=1750 nM) in rat brain membranes as measured by the displacement of [3H]clonidine[1].
Medetomidine (0.1-100 nM) inhibits the twitch response in field-stimulated mouse vas deferens, with a pD2 of 9.0[1].
In Vivo:Medetomidine (10-100 μg/kg; i.v. at 5-min intervals) produces a dose-dependent pupillary dilatation in pentobarbitone-anaesthetized rats[1].
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