VU0469650
CAS No. : 1443748-47-7
| Size | Price | Stock |
|---|---|---|
| 5mg | $156 | In-stock |
| 10mg | $235 | In-stock |
| 25mg | $470 | In-stock |
| 50mg | $700 | In-stock |
| 100mg | $1036 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-110191 |
| M.Wt: | 364.48 |
| Formula: | C22H28N4O |
| Purity: | >98 % |
| Solubility: | DMSO : 41.67 mg/mL (ultrasonic;warming;heat to 60°C) |
VU0469650 is a potent, selective and brain-penetrant negative allosteric modulator of mGlu1 receptor, with an IC50 of 99 nM[1].
IC50 & Target:IC50: 99 nM (mGlu1)[1]
In Vivo:VU0469650 (male Sprague-Dawley rats, 0.2 mg/kg, IV, once) exhibits moderate to high clearance, a moderate volume of distribution, and a half-life of approximately 1 hour[1].
VU0469650 (male Sprague-Dawley rats, 10 mg/kg, IP, once) shows an excellent selectivity profile and good exposure in both plasma and brain samples[1].
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