Deltarasin
CAS No. : 1440898-61-2
| Size | Price | Stock |
|---|---|---|
| 2mg | $60 | In-stock |
| 5mg | $120 | In-stock |
| 10mg | $200 | In-stock |
| 25mg | $360 | In-stock |
| 50mg | $540 | In-stock |
| 100mg | $810 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-15747 |
| M.Wt: | 603.75 |
| Formula: | C40H37N5O |
| Purity: | >98 % |
| Solubility: | H2O : 1 mg/mL (ultrasonic;warming;heat to 60°C);DMSO : 12.5 mg/mL (ultrasonic;warming;heat to 60°C) |
Deltarasin is an inhibitor of?KRAS-PDEδ interaction with?Kd?of 38 nM for binding to purified PDEδ. IC50 & Target: Kd: 38 nM (PDEδ) In Vitro: In liver cells, deltarasin inhibits the interaction of RAS with PDEδ with Kd?of 41 nM. Inhibition of PDEδ-KRAS interaction by deltarasin suppresses proliferation of human pancreatic ductal adenocarcinoma cells that are dependent on oncogenic KRAS[1]. In Vivo: Deltarasin (10 mg/kg, i.p.) impairs dose-dependent tumor growth in nude mice bearing subcutaneous human Panc-Tu-I tumour cell xenografts[1].
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