CB1-IN-1


CAS No. : 1429239-98-4

(Synonyms: BPRCB1184)

1429239-98-4
Price and Availability of CAS No. : 1429239-98-4
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5mg $420 In-stock
10mg $600 In-stock
50mg $1800 In-stock
100mg $2520 In-stock
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Cat. No. : HY-12790
M.Wt: 751.67
Formula: C33H31Cl2F3N6O3S2
Purity: >98 %
Solubility: DMSO : 125 mg/mL (ultrasonic)
Introduction of 1429239-98-4 :

CB1-IN-1 (BPRCB1184) is a peripherally restricted CB1R antagonist, with Ki of 0.3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively. IC50 value: 0.3 nM (Ki, CB1R) 21 nM (Ki, CB2R) Target: CB1R in vivo: CB1-IN-1 is a novel peripherally restricted cannabinoid 1 receptor antagonist with significant weight-loss efficacy in diet-induced obese mice. CB1-IN-1 has great potential to ameliorate this related metabolic syndrome.

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