C-82
CAS No. : 1422253-37-9
| Size | Price | Stock |
|---|---|---|
| 1mg | $110 | In-stock |
| 5mg | $470 | In-stock |
| 10mg | $835 | In-stock |
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| 100 mg | Get quote | |
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| Cat. No. : | HY-112359 |
| M.Wt: | 578.66 |
| Formula: | C33H34N6O4 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
C-82 is a second-generation specific CBP/β-catenin antagonist, which inhibits the binding between β-catenin and CBP and increases the binding between β-catenin and p300[1]. IC50 & Target:CBP/β-catenin[1] In Vitro:C-82 is an active form of PRI-724. C-82 inhibits the activation of isolated primary mouse quiescent hepatic stellate cells (HSCs) and promotes cell death in culture-activated HSCs[1]. In Vivo:PRI-724 is phosphorylated-C-82 and is rapidly hydrolyzed to its active form C-82 in vivo, and pre-clinical studies have shown a very acceptable toxicity profile[1].
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