GSK2798745
CAS No. : 1419609-94-1
| Size | Price | Stock |
|---|---|---|
| 5mg | $695 | In-stock |
| 10mg | $1250 | In-stock |
| 50mg | $2980 | In-stock |
| 100 mg | Get quote | |
| 200 mg | Get quote | |
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| Cat. No. : | HY-19765 |
| M.Wt: | 460.53 |
| Formula: | C25H28N6O3 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 100 mg/mL |
GSK2798745 is a potent, selective, and orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively. GSK2798745 can be used in cardiac and respiratory diseases research[1][2][3]. IC50 & Target: IC50: 1.8 nM (hTRPV4) and 1.6 nM (rTRPV4)[2] In Vitro: GSK2798745 inhibits TRPV4 agonist-induced impedance reduction in human umbilical vein endothelial cells (HUVECs)[3]. In Vivo: GSK2798745 inhibits TRPV4 agonist-mediated lung edema in rats in a dose-dependent manner[3].
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