FMK-MEA
CAS No. : 1414811-15-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $650 | In-stock |
| 10mg | $1040 | In-stock |
| 25mg | $2080 | In-stock |
| 50mg | $3328 | In-stock |
| 100mg | $5325 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-52101C |
| M.Wt: | 399.46 |
| Formula: | C21H26FN5O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor. IC50 & Target:p90 RSK[1] In Vitro: FMK-MEA is a water-soluble derivative of fmk. FMK-MEA treatment inhibits RSK2 kinase activity in diverse, highly invasive human cancer cell lines including 212LN, M4e, A549, and SKBR3 cells. Treatment with the RSK-specific inhibitor FMK-MEA significantly attenuates RSK2 activity, as assessed by the phosphorylation levels of Ser-386 and the consequent invasive ability of A549 cells[1]. In Vivo: FMK-MEA treatment (80 mg/kg/day for 16 days by intraperitoneal injection) in highly metastatic M4e cell xenograft nude mice results in a significant attenuation of LN metastasis. FMK-MEA treatment has no effect on the tumor size, and the proliferation rate of the primary tumor[1].
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