| Size | Price | Stock |
|---|---|---|
| 100 mg | Get quote | |
| 250 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-120291 |
| M.Wt: | 498.40 |
| Formula: | C25H25Cl2N5O2 |
| Purity: | >98 % |
| Solubility: |
ASP9436 is an orally active and blood-brain barrier permeable PDE10A inhibitor with an IC50 of 8 nM against human PDE10A. ASP9436 attenuates locomotor activity in mouse hyperactivity models and ameliorates visual recognition memory impairment in neonatal mice. ASP9436 is applicable to research related to schizophrenia[1]. In Vivo:ASP9436 (Compound 38 b) (0.001-30 mg/kg, p.o., single administration) attenuates locomotor activity and ameliorates visual recognition memory impairment in neonatal mice in the phencyclidine (PCP)-induced hyperlocomotion mouse model[1].
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