CGP52432
CAS No. : 139667-74-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $99 | In-stock |
| 10mg | $176 | In-stock |
| 25mg | $325 | In-stock |
| 50mg | $488 | In-stock |
| 100mg | $730 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-103531 |
| M.Wt: | 384.24 |
| Formula: | C15H24Cl2NO4P |
| Purity: | >98 % |
| Solubility: | DMSO : 5 mg/mL (ultrasonic;warming);H2O : 4 mg/mL (ultrasonic;warming;heat to 60°C) |
CGP52432 is a GABAB receptor antagonist, with an IC50 of 85 nM. IC50 & Target: IC50: 85 nM (GABAB receptor)[1] In Vitro: CGP52432 is a GABAB receptor antagonist, with an IC50 of 85 nM, 35- and 100-fold lower than at the receptors regulating somatostatin and glutamate overflow, respectively[1]. In Vivo: CGP52432 (10, 30 mg/kg) shows no effect on the total arm entries and total head dips of mice on the elevated-plus maze[2]. CGP52432 (100 nmol/kg, i.v., or 1 nmol/kg, i.c.v.) abolishes the suppressive effects of GABA ( 50 μmol/kg, i.v.) on enhanced renal sympathetic nerve activity (RSNA) during ischaemia, causeing elimination of the renoprotective effects of GABA in rats[3].
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